NA-DB

Compound Info

NAs

Base Info

Cluster

Name

Target

MolWt

NAs.002742

GW813360X

Target name	Tax id
Casein kinase I alpha	7054.0
MAP kinase p38 delta	7054.0
PI4-kinase beta subunit	7054.0
Serine/threonine-protein kinase Aurora-B	7054.0
Cyclin-dependent kinase 2	7054.0
Fibroblast growth factor receptor 4	7054.0
Renilla-luciferin 2-monooxygenase	7054.0
Protein kinase C eta	7054.0
Tyrosine-protein kinase BLK	7054.0
Tyrosine-protein kinase JAK2	7054.0
Tyrosine-protein kinase receptor UFO	7054.0
Fibroblast growth factor receptor 1	7054.0
Protein tyrosine kinase 2 beta	7054.0
Ribosomal protein S6 kinase 1	7054.0
Proto-oncogene tyrosine-protein kinase ROS	7054.0
Tyrosine-protein kinase receptor RET	7054.0
Tyrosine-protein kinase JAK3	7054.0
Vascular endothelial growth factor receptor 2	7054.0
Casein kinase I isoform gamma-3	7054.0
Tyrosine-protein kinase HCK	7054.0
Maternal embryonic leucine zipper kinase	7054.0
Phosphorylase kinase gamma subunit 2	7054.0
cGMP-dependent protein kinase 2	7054.0
MAP kinase ERK2	7054.0
Serine/threonine-protein kinase DCLK2	7054.0
Ribosomal protein S6 kinase alpha 5	7054.0
Inhibitor of nuclear factor kappa B kinase beta subunit	7054.0
Mitogen-activated protein kinase kinase kinase kinase 2	7054.0
Serine/threonine-protein kinase PAK 2	7054.0
MAP kinase-activated protein kinase 3	7054.0
Death-associated protein kinase 1	7054.0
CaM kinase I delta	7054.0
Inhibitor of nuclear factor kappa B kinase alpha subunit	7054.0
Tyrosine-protein kinase LCK	7054.0
Serine/threonine-protein kinase RAF	7054.0
Serine/threonine-protein kinase PIM1	7054.0
3-phosphoinositide dependent protein kinase-1	7054.0
Insulin receptor-related protein	7054.0
Serine/threonine-protein kinase MRCK beta	7054.0
MAP kinase-activated protein kinase 5	7054.0
Fibroblast growth factor receptor 2	7054.0
Rho-associated protein kinase 2	7054.0
Vascular endothelial growth factor receptor 3	7054.0
Epidermal growth factor receptor erbB1	7054.0
Serine/threonine-protein kinase c-TAK1	7054.0
Protein kinase C mu	7054.0
Serine/threonine-protein kinase PRKX	7054.0
MAP kinase ERK1	7054.0
Serine/threonine-protein kinase PIM2	7054.0
Leukocyte tyrosine kinase receptor	7054.0
Ephrin type-A receptor 2	7054.0
Tyrosine kinase non-receptor protein 2	7054.0
Pyruvate dehydrogenase kinase isoform 1	7054.0
cGMP-dependent protein kinase 1 beta	7054.0
Protein kinase C gamma	7054.0
Tyrosine-protein kinase Lyn	7054.0
Serine/threonine-protein kinase D2	7054.0
Inhibitor of nuclear factor kappa B kinase epsilon subunit	7054.0
Ephrin type-A receptor 4	7054.0
Leucine-rich repeat serine/threonine-protein kinase 2	7054.0
MAP kinase signal-integrating kinase 2	7054.0
MAP kinase p38 alpha	7054.0
Ribosomal protein S6 kinase alpha 1	7054.0
Homeodomain-interacting protein kinase 4	7054.0
Dual specificity mitogen-activated protein kinase kinase 1	7054.0
Serine/threonine-protein kinase AKT	7054.0
Protein kinase C nu	7054.0
Dual specificity protein kinase CLK3	7054.0
Serine/threonine-protein kinase PIM3	7054.0
Tyrosine-protein kinase BMX	7054.0
BR serine/threonine-protein kinase 1	7054.0
Serine/threonine-protein kinase SRPK3	7054.0
CDK3/Cyclin E	7054.0
Serine/threonine-protein kinase PLK1	7054.0
Serine/threonine-protein kinase B-raf	7054.0
CaM kinase II alpha	7054.0
Serine/threonine-protein kinase Aurora-A	7054.0
MAP kinase-activated protein kinase 2	7054.0
Tyrosine-protein kinase TXK	7054.0
AMP-activated protein kinase	7054.0
alpha-1 subunit	7054.0
Serine/threonine-protein kinase Sgk2	7054.0
Tyrosine-protein kinase FER	7054.0
Discoidin domain-containing receptor 2	7054.0
AMP-activated protein kinase	7054.0
alpha-2 subunit	7054.0
ALK tyrosine kinase receptor	7054.0
Muscle	7054.0
skeletal receptor tyrosine protein kinase	7054.0
Tyrosine-protein kinase FYN	7054.0
Receptor protein-tyrosine kinase erbB-4	7054.0
MAP/microtubule affinity-regulating kinase 4	7054.0
Protein kinase C theta	7054.0
Sphingosine kinase 2	7054.0
Tyrosine-protein kinase receptor FLT3	7054.0
Tyrosine-protein kinase ITK/TSK	7054.0
Serine/threonine-protein kinase Sgk3	7054.0
Tyrosine-protein kinase FRK	7054.0
CaM kinase II delta	7054.0
Serine/threonine-protein kinase SIK1	7054.0
Tyrosine-protein kinase CSK	7054.0
Serine/threonine-protein kinase AKT2	7054.0
CaM kinase IV	7054.0
Insulin-like growth factor I receptor	7054.0
Tyrosine-protein kinase ZAP-70	7054.0
MAP/microtubule affinity-regulating kinase 2	7054.0
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	7054.0
Neurotrophic tyrosine kinase receptor type 2	7054.0
Serine/threonine-protein kinase Nek1	7054.0
Serine/threonine-protein kinase PAK6	7054.0
Tyrosine-protein kinase YES	7054.0
Serine/threonine-protein kinase NEK2	7054.0
Macrophage-stimulating protein receptor	7054.0
Serine/threonine-protein kinase MST2	7054.0
Serine/threonine-protein kinase NEK6	7054.0
Tyrosine-protein kinase ABL2	7054.0
Serine/threonine-protein kinase MRCK-A	7054.0
Ribosomal protein S6 kinase alpha 3	7054.0
Dual specificity protein kinase TTK	7054.0
Serine/threonine-protein kinase MARK1	7054.0
Tyrosine-protein kinase SYK	7054.0
Tyrosine-protein kinase ABL	7054.0
Tyrosine-protein kinase receptor TYRO3	7054.0
Casein kinase I gamma 2	7054.0
PI3-kinase p110-delta subunit	7054.0
Tyrosine-protein kinase JAK1	7054.0
PI3-kinase p110-alpha subunit	7054.0
Tyrosine-protein kinase FES	7054.0
Cyclin-dependent kinase 6	7054.0
Fibroblast growth factor receptor 3	7054.0
Tyrosine-protein kinase Srms	7054.0
Casein kinase I gamma 1	7054.0
Protein kinase C beta	7054.0
Serine/threonine-protein kinase NEK9	7054.0
MAP kinase-interacting serine/threonine-protein kinase MNK1	7054.0
Testis-specific serine/threonine-protein kinase 2	7054.0
Serine/threonine-protein kinase 10	7054.0
Glycogen synthase kinase-3 beta	7054.0
Tyrosine-protein kinase BTK	7054.0
Platelet-derived growth factor receptor alpha	7054.0
Glycogen synthase kinase-3	7054.0
Dual-specificity tyrosine-phosphorylation regulated kinase 1A	7054.0
MAP kinase p38 beta	7054.0
BR serine/threonine-protein kinase 2	7054.0
Cyclin-dependent kinase 5	7054.0
Tyrosine-protein kinase BRK	7054.0
Proto-oncogene tyrosine-protein kinase MER	7054.0
Serine/threonine-protein kinase PAK 3	7054.0
G protein-coupled receptor kinase 7	7054.0
Rho-associated protein kinase 1	7054.0
Protein kinase C alpha	7054.0
Ephrin type-B receptor 4	7054.0
Protein kinase C iota	7054.0
Interleukin-1 receptor-associated kinase 4	7054.0
Ephrin type-B receptor 2	7054.0
MAP kinase p38 gamma	7054.0
Ribosomal protein S6 kinase alpha 2	7054.0
Testis-specific serine/threonine-protein kinase 1	7054.0
c-Jun N-terminal kinase 2	7054.0
Ribosomal protein S6 kinase alpha 6	7054.0
NT-3 growth factor receptor	7054.0
Insulin receptor	7054.0
Dual-specificity tyrosine-phosphorylation regulated kinase 2	7054.0
Serine/threonine-protein kinase PAK 1	7054.0
Stem cell growth factor receptor	7054.0
Tyrosine-protein kinase TYK2	7054.0
Non-receptor tyrosine-protein kinase TNK1	7054.0
Hepatocyte growth factor receptor	7054.0
Cyclin-dependent kinase 4	7054.0
Dual specificity protein kinase CLK2	7054.0
Serine/threonine-protein kinase MST1	7054.0
Glycogen synthase kinase-3 alpha	7054.0
Serine/threonine-protein kinase PAK7	7054.0
Ephrin type-A receptor 3	7054.0
Platelet-derived growth factor receptor beta	7054.0
Serine/threonine-protein kinase NEK7	7054.0
G protein-coupled receptor kinase 6	7054.0
Sphingosine kinase 1	7054.0
Ephrin type-B receptor 3	7054.0
Homeodomain-interacting protein kinase 1	7054.0
Misshapen-like kinase 1	7054.0
Tyrosine-protein kinase FGR	7054.0
Casein kinase II alpha	7054.0
Tyrosine-protein kinase TEC	7054.0
Serine/threonine-protein kinase MST4	7054.0
Cyclin-dependent kinase 1	7054.0
Phosphorylase kinase gamma subunit 1	7054.0
Macrophage colony stimulating factor receptor	7054.0
Receptor protein-tyrosine kinase erbB-2	7054.0
Ribosomal protein S6 kinase alpha 4	7054.0
Serine/threonine-protein kinase SRPK1	7054.0
Serine/threonine-protein kinase TBK1	7054.0
Serine/threonine-protein kinase AKT3	7054.0
Vascular endothelial growth factor receptor 1	7054.0
Serine/threonine-protein kinase Aurora-C	7054.0
Tyrosine-protein kinase SRC	7054.0
Tyrosine-protein kinase TIE-2	7054.0
Nerve growth factor receptor Trk-A	7054.0
PAS domain-containing serine/threonine-protein kinase	7054.0
Serine/threonine-protein kinase SIK2	7054.0
NUAK family SNF1-like kinase 1	7054.0
cAMP-dependent protein kinase alpha-catalytic subunit	7054.0
Serine/threonine-protein kinase Chk1	7054.0
Serine/threonine-protein kinase Sgk1	7054.0
Serine/threonine-protein kinase Chk2	7054.0
Mitogen-activated protein kinase kinase kinase kinase 4	7054.0
Luciferin 4-monooxygenase	7054.0

345.366

Chemical Representations
InChI	InChI=1S/C18H15N7O/c1-26-15-4-2-3-14(9-15)25-12-22-16-17(20-11-21-18(16)25)24-23-10-13-5-7-19-8-6-13/h2-12H,1H3,(H,20,21,24)/b23-10+
InChI Key	VARGUUBRJVQGHK-AUEPDCJTSA-N
SMILES	COc1cccc(-n2cnc3c(N/N=C/c4ccncc4)ncnc32)c1
Molecular Formula	C18H15N7O

Functional Fragments
Base	Ribose	Phosphate
Unmatch	Match

Calculated Properties
logP	2.665	Computed by RDKit
Heavy Atom Count	26	Computed by RDKit
Ring Count	4	Computed by RDKit
Hydrogen Bond Acceptor Count	8	Computed by RDKit
Hydrogen Bond Donor Count	1	Computed by RDKit
Rotatable Bond Count	5	Computed by RDKit
Topological Polar Surface Area	90.110	Computed by RDKit

Activity Data
Target	Activity type	Relation	Value	Unit	Assay	Source
Glycogen synthase kinase-3	IC50	=	630.96	nM	Inhibition of GSK3	CHEMBL1146115
Serine/threonine-protein kinase AKT	Inhibition	=	-4.15	%	GSK_PKIS: AKT1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase AKT2	Inhibition	=	-3.57	%	GSK_PKIS: AKT2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase AKT3	Inhibition	=	-4.17	%	GSK_PKIS: AKT3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
G protein-coupled receptor kinase 6	Inhibition	=	2.45	%	GSK_PKIS: GRK6 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
G protein-coupled receptor kinase 7	Inhibition	=	1.71	%	GSK_PKIS: GRK7 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MRCK-A	Inhibition	=	1.59	%	GSK_PKIS: MRCKA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MRCK beta	Inhibition	=	0.38	%	GSK_PKIS: MRCKB mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 5	Inhibition	=	-0.31	%	GSK_PKIS: MSK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 4	Inhibition	=	2.44	%	GSK_PKIS: MSK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase 1	Inhibition	=	-0.32	%	GSK_PKIS: p70s6K1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
3-phosphoinositide dependent protein kinase-1	Inhibition	=	0.77	%	GSK_PKIS: PDK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
cAMP-dependent protein kinase alpha-catalytic subunit	Inhibition	=	-1.92	%	GSK_PKIS: PKA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C alpha	Inhibition	=	-2.58	%	GSK_PKIS: PKC-alpha mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C beta	Inhibition	=	3.24	%	GSK_PKIS: PKC-beta1 (splice variant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C eta	Inhibition	=	3.47	%	GSK_PKIS: PKC-eta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C gamma	Inhibition	=	0.93	%	GSK_PKIS: PKC-gamma mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C iota	Inhibition	=	0.58	%	GSK_PKIS: PKC-iota mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C theta	Inhibition	=	0.62	%	GSK_PKIS: PKC-theta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C beta	Inhibition	=	2.34	%	GSK_PKIS: PKC-beta2 (splice variant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C mu	Inhibition	=	-2.1	%	GSK_PKIS: PRKD1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase D2	Inhibition	=	-4.34	%	GSK_PKIS: PRKD2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C nu	Inhibition	=	-3.34	%	GSK_PKIS: PRKD3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
cGMP-dependent protein kinase 1 beta	Inhibition	=	0.67	%	GSK_PKIS: PRKG1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
cGMP-dependent protein kinase 2	Inhibition	=	3.29	%	GSK_PKIS: PRKG2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PRKX	Inhibition	=	1.92	%	GSK_PKIS: PRKX mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Rho-associated protein kinase 1	Inhibition	=	0.59	%	GSK_PKIS: ROCK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Rho-associated protein kinase 2	Inhibition	=	3.27	%	GSK_PKIS: ROCK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 1	Inhibition	=	2.62	%	GSK_PKIS: RSK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 3	Inhibition	=	2.12	%	GSK_PKIS: RSK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 2	Inhibition	=	-0.37	%	GSK_PKIS: RSK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 6	Inhibition	=	-0.06	%	GSK_PKIS: RSK4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk1	Inhibition	=	1.3	%	GSK_PKIS: SGK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk2	Inhibition	=	1.67	%	GSK_PKIS: SGK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk3	Inhibition	=	3.19	%	GSK_PKIS: SGK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
AMP-activated protein kinase, alpha-1 subunit	Inhibition	=	1.05	%	GSK_PKIS: AMPKA1 (A1B1G1) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
AMP-activated protein kinase, alpha-2 subunit	Inhibition	=	-1.1	%	GSK_PKIS: AMPKA2 (A2B1G1) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
NUAK family SNF1-like kinase 1	Inhibition	=	2.39	%	GSK_PKIS: ARK5 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
BR serine/threonine-protein kinase 1	Inhibition	=	-0.01	%	GSK_PKIS: BRSK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
BR serine/threonine-protein kinase 2	Inhibition	=	-0.23	%	GSK_PKIS: BRSK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
CaM kinase I delta	Inhibition	=	0.54	%	GSK_PKIS: CAMK1D mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
CaM kinase II alpha	Inhibition	=	0.58	%	GSK_PKIS: CAMK2A mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
CaM kinase II delta	Inhibition	=	-1.07	%	GSK_PKIS: CAMK2D mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
CaM kinase IV	Inhibition	=	-2.88	%	GSK_PKIS: CAMK4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Chk1	Inhibition	=	0.34	%	GSK_PKIS: CHEK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Chk2	Inhibition	=	-0.94	%	GSK_PKIS: CHEK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Death-associated protein kinase 1	Inhibition	=	-0.67	%	GSK_PKIS: DAPK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase DCLK2	Inhibition	=	-3.07	%	GSK_PKIS: DCAMKL2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 2	Inhibition	=	-0.39	%	GSK_PKIS: MAPKAPK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 3	Inhibition	=	-0.9	%	GSK_PKIS: MAPKAPK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MARK1	Inhibition	=	1.01	%	GSK_PKIS: MARK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase c-TAK1	Inhibition	=	1.08	%	GSK_PKIS: MARK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP/microtubule affinity-regulating kinase 4	Inhibition	=	0.84	%	GSK_PKIS: MARK4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Maternal embryonic leucine zipper kinase	Inhibition	=	-1.92	%	GSK_PKIS: MELK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-interacting serine/threonine-protein kinase MNK1	Inhibition	=	0.43	%	GSK_PKIS: MKNK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase signal-integrating kinase 2	Inhibition	=	3.13	%	GSK_PKIS: MNK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP/microtubule affinity-regulating kinase 2	Inhibition	=	0.99	%	GSK_PKIS: PAR-1Balpha mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
PAS domain-containing serine/threonine-protein kinase	Inhibition	=	1.87	%	GSK_PKIS: PASK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Phosphorylase kinase gamma subunit 1	Inhibition	=	-0.02	%	GSK_PKIS: PHKG1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Phosphorylase kinase gamma subunit 2	Inhibition	=	1.83	%	GSK_PKIS: PHKG2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM1	Inhibition	=	-0.24	%	GSK_PKIS: PIM1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM2	Inhibition	=	-3.51	%	GSK_PKIS: PIM2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM3	Inhibition	=	3.67	%	GSK_PKIS: PIM3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 5	Inhibition	=	0.59	%	GSK_PKIS: PRAK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SIK1	Inhibition	=	1.88	%	GSK_PKIS: SNF1LK (SIK) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SIK2	Inhibition	=	9.07	%	GSK_PKIS: SNF1LK2 (QIK) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase TBK1	Inhibition	=	0.99	%	GSK_PKIS: TBK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Testis-specific serine/threonine-protein kinase 1	Inhibition	=	0.41	%	GSK_PKIS: TSSK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Testis-specific serine/threonine-protein kinase 2	Inhibition	=	0.37	%	GSK_PKIS: TSSK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I alpha	Inhibition	=	0.17	%	GSK_PKIS: CK1a mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I gamma 1	Inhibition	=	-3.8	%	GSK_PKIS: CK1-g1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I gamma 2	Inhibition	=	-3.36	%	GSK_PKIS: CK1-g2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I isoform gamma-3	Inhibition	=	-3.39	%	GSK_PKIS: CK1-g3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 1	Inhibition	=	-3.5	%	GSK_PKIS: CDK1/cyclinB mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 2	Inhibition	=	-3.99	%	GSK_PKIS: CDK2/cyclinA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 2	Inhibition	=	-3.22	%	GSK_PKIS: CDK2/cyclinE mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
CDK3/Cyclin E	Inhibition	=	-0.66	%	GSK_PKIS: CDK3/cyclinE mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 4	Inhibition	=	-6.94	%	GSK_PKIS: CDK4/cyclinD mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 5	Inhibition	=	-3.69	%	GSK_PKIS: CDK5/p35 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 6	Inhibition	=	-0.76	%	GSK_PKIS: CDK6/cyclinD3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase CLK2	Inhibition	=	3.04	%	GSK_PKIS: CLK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase CLK3	Inhibition	=	-3.93	%	GSK_PKIS: CLK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Inhibition	=	-3.39	%	GSK_PKIS: DYRK1A mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Inhibition	=	-3.26	%	GSK_PKIS: DYRK1B mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual-specificity tyrosine-phosphorylation regulated kinase 2	Inhibition	=	0.79	%	GSK_PKIS: DYRK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Glycogen synthase kinase-3 alpha	Inhibition	=	3.64	%	GSK_PKIS: GSK3A mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Glycogen synthase kinase-3 beta	Inhibition	=	3.02	%	GSK_PKIS: GSK3B mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Homeodomain-interacting protein kinase 1	Inhibition	=	-2.33	%	GSK_PKIS: HIPK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Homeodomain-interacting protein kinase 4	Inhibition	=	-0.66	%	GSK_PKIS: HIPK4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
c-Jun N-terminal kinase 2	Inhibition	=	-1.67	%	GSK_PKIS: JNK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase ERK2	Inhibition	=	-1.43	%	GSK_PKIS: MAPK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase ERK1	Inhibition	=	0.83	%	GSK_PKIS: MAPK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SRPK3	Inhibition	=	-0.93	%	GSK_PKIS: MSSK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 alpha	Inhibition	=	2.63	%	GSK_PKIS: P38alpha mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 beta	Inhibition	=	1.35	%	GSK_PKIS: P38beta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 delta	Inhibition	=	-0.64	%	GSK_PKIS: P38delta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 gamma	Inhibition	=	-1.4	%	GSK_PKIS: P38gamma mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SRPK1	Inhibition	=	1.41	%	GSK_PKIS: SRPK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
PI3-kinase p110-alpha subunit	Inhibition	=	-0.19	%	GSK_PKIS: PI3K-alpha mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
PI3-kinase p110-delta subunit	Inhibition	=	-1.29	%	GSK_PKIS: PI3K-delta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
PI4-kinase beta subunit	Inhibition	=	5.84	%	GSK_PKIS: PI4K-beta mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Sphingosine kinase 1	Inhibition	=	-0.37	%	GSK_PKIS: SPHK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Sphingosine kinase 2	Inhibition	=	0.58	%	GSK_PKIS: SPHK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Casein kinase II alpha	Inhibition	=	0.97	%	GSK_PKIS: CK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase alpha subunit	Inhibition	=	0.84	%	GSK_PKIS: IKKA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase beta subunit	Inhibition	=	1.12	%	GSK_PKIS: IKKB mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase epsilon subunit	Inhibition	=	3.81	%	GSK_PKIS: IKKE mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Nek1	Inhibition	=	0.0	%	GSK_PKIS: NEK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK2	Inhibition	=	-1.74	%	GSK_PKIS: NEK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK6	Inhibition	=	2.37	%	GSK_PKIS: NEK6 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK7	Inhibition	=	-0.81	%	GSK_PKIS: NEK7 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK9	Inhibition	=	0.98	%	GSK_PKIS: NEK9 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PLK1	Inhibition	=	-1.9	%	GSK_PKIS: PLK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase TTK	Inhibition	=	0.25	%	GSK_PKIS: TTK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-A	Inhibition	=	-0.8	%	GSK_PKIS: Aurora-A mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-B	Inhibition	=	0.64	%	GSK_PKIS: Aurora-B mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-C	Inhibition	=	0.73	%	GSK_PKIS: Aurora-C mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase 10	Inhibition	=	4.49	%	GSK_PKIS: LOK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Mitogen-activated protein kinase kinase kinase kinase 2	Inhibition	=	1.19	%	GSK_PKIS: MAP4K2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Mitogen-activated protein kinase kinase kinase kinase 4	Inhibition	=	1.22	%	GSK_PKIS: MAP4K4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Dual specificity mitogen-activated protein kinase kinase 1	Inhibition	=	-0.13	%	GSK_PKIS: MEK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Misshapen-like kinase 1	Inhibition	=	2.27	%	GSK_PKIS: MINK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST1	Inhibition	=	3.6	%	GSK_PKIS: MST1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST2	Inhibition	=	4.46	%	GSK_PKIS: MST2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST4	Inhibition	=	0.98	%	GSK_PKIS: MST4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 1	Inhibition	=	2.37	%	GSK_PKIS: PAK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 2	Inhibition	=	-1.03	%	GSK_PKIS: PAK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 3	Inhibition	=	-1.14	%	GSK_PKIS: PAK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK7	Inhibition	=	6.09	%	GSK_PKIS: PAK5 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK6	Inhibition	=	5.99	%	GSK_PKIS: PAK6 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	30.77	%	GSK_PKIS: ABL1 (E255K mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	47.15	%	GSK_PKIS: ABL1 (H396P mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	44.72	%	GSK_PKIS: ABL1 (M351T mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	40.08	%	GSK_PKIS: ABL1 (Q252H mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	1.94	%	GSK_PKIS: ABL1 (T315I mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	44.65	%	GSK_PKIS: ABL1 (Y253F mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	28.96	%	GSK_PKIS: ABL1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
ALK tyrosine kinase receptor	Inhibition	=	-1.9	%	GSK_PKIS: ALK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL2	Inhibition	=	12.69	%	GSK_PKIS: ARG mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor UFO	Inhibition	=	3.99	%	GSK_PKIS: AXL mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BLK	Inhibition	=	-0.3	%	GSK_PKIS: BLK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BMX	Inhibition	=	-0.75	%	GSK_PKIS: BMX mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BRK	Inhibition	=	0.43	%	GSK_PKIS: BRK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BTK	Inhibition	=	-2.61	%	GSK_PKIS: BTK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase CSK	Inhibition	=	1.91	%	GSK_PKIS: CSK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Discoidin domain-containing receptor 2	Inhibition	=	-0.19	%	GSK_PKIS: DDR2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	2.02	%	GSK_PKIS: EGFR mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	5.72	%	GSK_PKIS: EGFR (L858R mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	1.61	%	GSK_PKIS: EGFR (L861Q mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	-0.92	%	GSK_PKIS: EGFR (T790M mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	-1.35	%	GSK_PKIS: EGFR (T790M-L858R mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 2	Inhibition	=	-0.82	%	GSK_PKIS: EPHA2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 3	Inhibition	=	-3.39	%	GSK_PKIS: EPHA3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 4	Inhibition	=	3.18	%	GSK_PKIS: EPHA4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 2	Inhibition	=	2.42	%	GSK_PKIS: EPHB2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 3	Inhibition	=	-8.69	%	GSK_PKIS: EPHB3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 4	Inhibition	=	-2.1	%	GSK_PKIS: EPHB4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Receptor protein-tyrosine kinase erbB-2	Inhibition	=	0.94	%	GSK_PKIS: ERBB2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Receptor protein-tyrosine kinase erbB-4	Inhibition	=	-3.73	%	GSK_PKIS: ERBB4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FER	Inhibition	=	4.18	%	GSK_PKIS: FER mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FES	Inhibition	=	-0.04	%	GSK_PKIS: FES mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 1	Inhibition	=	-7.19	%	GSK_PKIS: FGFR1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 2	Inhibition	=	-3.25	%	GSK_PKIS: FGFR2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 3	Inhibition	=	-3.58	%	GSK_PKIS: FGFR3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 4	Inhibition	=	-4.06	%	GSK_PKIS: FGFR4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FGR	Inhibition	=	6.79	%	GSK_PKIS: FGR mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 1	Inhibition	=	-1.12	%	GSK_PKIS: FLT1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor FLT3	Inhibition	=	0.88	%	GSK_PKIS: FLT3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor FLT3	Inhibition	=	7.7	%	GSK_PKIS: FLT3 (D835Y mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 3	Inhibition	=	-13.03	%	GSK_PKIS: FLT4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Macrophage colony stimulating factor receptor	Inhibition	=	4.43	%	GSK_PKIS: FMS mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FYN	Inhibition	=	-0.06	%	GSK_PKIS: FYN mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase HCK	Inhibition	=	0.9	%	GSK_PKIS: HCK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Insulin-like growth factor I receptor	Inhibition	=	-11.38	%	GSK_PKIS: IGF1R mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Insulin receptor	Inhibition	=	-2.78	%	GSK_PKIS: INSR mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Insulin receptor-related protein	Inhibition	=	1.0	%	GSK_PKIS: IRR mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ITK/TSK	Inhibition	=	-2.76	%	GSK_PKIS: ITK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK1	Inhibition	=	4.44	%	GSK_PKIS: JAK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK2	Inhibition	=	0.27	%	GSK_PKIS: JAK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK3	Inhibition	=	-2.48	%	GSK_PKIS: JAK3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 2	Inhibition	=	-0.11	%	GSK_PKIS: KDR mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	33.37	%	GSK_PKIS: KIT mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	0.1	%	GSK_PKIS: KIT (D816V mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	-2.23	%	GSK_PKIS: KIT (T6701 mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	3.15	%	GSK_PKIS: KIT (V560G mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase LCK	Inhibition	=	3.69	%	GSK_PKIS: LCK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Leukocyte tyrosine kinase receptor	Inhibition	=	-1.69	%	GSK_PKIS: LTK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Lyn	Inhibition	=	7.17	%	GSK_PKIS: LYN A (splice variant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Lyn	Inhibition	=	6.07	%	GSK_PKIS: LYN B (splice variant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Proto-oncogene tyrosine-protein kinase MER	Inhibition	=	0.12	%	GSK_PKIS: MER mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Hepatocyte growth factor receptor	Inhibition	=	0.87	%	GSK_PKIS: MET mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Muscle, skeletal receptor tyrosine protein kinase	Inhibition	=	2.4	%	GSK_PKIS: MUSK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	17.93	%	GSK_PKIS: PDGFRA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	4.61	%	GSK_PKIS: PDGFRA (D842V mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	2.14	%	GSK_PKIS: PDGFRA (T674I mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	10.33	%	GSK_PKIS: PDGFRA (V561D mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor beta	Inhibition	=	13.18	%	GSK_PKIS: PDGFRB mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FRK	Inhibition	=	-0.1	%	GSK_PKIS: PTK5 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Protein tyrosine kinase 2 beta	Inhibition	=	-4.12	%	GSK_PKIS: PYK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	3.89	%	GSK_PKIS: RET mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	-0.06	%	GSK_PKIS: RET (V804L mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	2.51	%	GSK_PKIS: RET (Y791F mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Macrophage-stimulating protein receptor	Inhibition	=	0.89	%	GSK_PKIS: RON mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Proto-oncogene tyrosine-protein kinase ROS	Inhibition	=	-1.03	%	GSK_PKIS: ROS mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase SRC	Inhibition	=	12.48	%	GSK_PKIS: SRC mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Srms	Inhibition	=	2.47	%	GSK_PKIS: SRMS mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase SYK	Inhibition	=	1.9	%	GSK_PKIS: SYK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TEC	Inhibition	=	-2.49	%	GSK_PKIS: TEC mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TIE-2	Inhibition	=	-0.9	%	GSK_PKIS: TIE2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Non-receptor tyrosine-protein kinase TNK1	Inhibition	=	1.98	%	GSK_PKIS: TNK1 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine kinase non-receptor protein 2	Inhibition	=	0.06	%	GSK_PKIS: TNK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Nerve growth factor receptor Trk-A	Inhibition	=	-1.67	%	GSK_PKIS: TRKA mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Neurotrophic tyrosine kinase receptor type 2	Inhibition	=	0.22	%	GSK_PKIS: TRKB mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
NT-3 growth factor receptor	Inhibition	=	0.58	%	GSK_PKIS: TRKC mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TXK	Inhibition	=	-1.8	%	GSK_PKIS: TXK mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TYK2	Inhibition	=	3.07	%	GSK_PKIS: TYK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor TYRO3	Inhibition	=	1.07	%	GSK_PKIS: TYRO3 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase YES	Inhibition	=	7.55	%	GSK_PKIS: YES mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ZAP-70	Inhibition	=	-2.42	%	GSK_PKIS: ZAP70 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase B-raf	Inhibition	=	-0.31	%	GSK_PKIS: BRAF mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase B-raf	Inhibition	=	-0.89	%	GSK_PKIS: BRAF (V599E mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase RAF	Inhibition	=	-3.41	%	GSK_PKIS: CRAF mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Interleukin-1 receptor-associated kinase 4	Inhibition	=	-2.35	%	GSK_PKIS: IRAK4 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Leucine-rich repeat serine/threonine-protein kinase 2	Inhibition	=	-1.76	%	GSK_PKIS: LRRK2 mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Leucine-rich repeat serine/threonine-protein kinase 2	Inhibition	=	0.11	%	GSK_PKIS: LRRK2 (G2019S mutant) mean inhibition at 0.1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase AKT	Inhibition	=	-3.41	%	GSK_PKIS: AKT1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase AKT2	Inhibition	=	-4.73	%	GSK_PKIS: AKT2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase AKT3	Inhibition	=	-3.32	%	GSK_PKIS: AKT3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
G protein-coupled receptor kinase 6	Inhibition	=	8.28	%	GSK_PKIS: GRK6 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
G protein-coupled receptor kinase 7	Inhibition	=	5.64	%	GSK_PKIS: GRK7 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MRCK-A	Inhibition	=	3.69	%	GSK_PKIS: MRCKA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MRCK beta	Inhibition	=	0.7	%	GSK_PKIS: MRCKB mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 5	Inhibition	=	1.02	%	GSK_PKIS: MSK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 4	Inhibition	=	3.95	%	GSK_PKIS: MSK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase 1	Inhibition	=	1.15	%	GSK_PKIS: p70s6K1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Pyruvate dehydrogenase kinase isoform 1	Inhibition	=	1.39	%	GSK_PKIS: PDK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
cAMP-dependent protein kinase alpha-catalytic subunit	Inhibition	=	0.18	%	GSK_PKIS: PKA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C alpha	Inhibition	=	-3.28	%	GSK_PKIS: PKC-alpha mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C beta	Inhibition	=	5.82	%	GSK_PKIS: PKC-beta1 (splice variant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C eta	Inhibition	=	0.69	%	GSK_PKIS: PKC-eta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C gamma	Inhibition	=	3.14	%	GSK_PKIS: PKC-gamma mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C iota	Inhibition	=	-0.97	%	GSK_PKIS: PKC-iota mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C theta	Inhibition	=	4.42	%	GSK_PKIS: PKC-theta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C beta	Inhibition	=	2.1	%	GSK_PKIS: PKC-beta2 (splice variant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C mu	Inhibition	=	-5.45	%	GSK_PKIS: PRKD1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase D2	Inhibition	=	-5.5	%	GSK_PKIS: PRKD2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein kinase C nu	Inhibition	=	-4.97	%	GSK_PKIS: PRKD3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
cGMP-dependent protein kinase 1 beta	Inhibition	=	3.77	%	GSK_PKIS: PRKG1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
cGMP-dependent protein kinase 2	Inhibition	=	4.98	%	GSK_PKIS: PRKG2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PRKX	Inhibition	=	5.16	%	GSK_PKIS: PRKX mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Rho-associated protein kinase 1	Inhibition	=	1.07	%	GSK_PKIS: ROCK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Rho-associated protein kinase 2	Inhibition	=	6.91	%	GSK_PKIS: ROCK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 1	Inhibition	=	4.66	%	GSK_PKIS: RSK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 3	Inhibition	=	4.76	%	GSK_PKIS: RSK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 2	Inhibition	=	0.82	%	GSK_PKIS: RSK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ribosomal protein S6 kinase alpha 6	Inhibition	=	1.9	%	GSK_PKIS: RSK4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk1	Inhibition	=	4.05	%	GSK_PKIS: SGK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk2	Inhibition	=	2.41	%	GSK_PKIS: SGK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Sgk3	Inhibition	=	3.83	%	GSK_PKIS: SGK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
AMP-activated protein kinase, alpha-1 subunit	Inhibition	=	3.79	%	GSK_PKIS: AMPKA1 (A1B1G1) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
AMP-activated protein kinase, alpha-2 subunit	Inhibition	=	1.47	%	GSK_PKIS: AMPKA2 (A2B1G1) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
NUAK family SNF1-like kinase 1	Inhibition	=	22.32	%	GSK_PKIS: ARK5 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
BR serine/threonine-protein kinase 1	Inhibition	=	4.34	%	GSK_PKIS: BRSK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
BR serine/threonine-protein kinase 2	Inhibition	=	6.3	%	GSK_PKIS: BRSK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
CaM kinase I delta	Inhibition	=	-0.39	%	GSK_PKIS: CAMK1D mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
CaM kinase II alpha	Inhibition	=	1.18	%	GSK_PKIS: CAMK2A mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
CaM kinase II delta	Inhibition	=	-1.61	%	GSK_PKIS: CAMK2D mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
CaM kinase IV	Inhibition	=	-5.3	%	GSK_PKIS: CAMK4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Chk1	Inhibition	=	0.31	%	GSK_PKIS: CHEK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Chk2	Inhibition	=	-0.32	%	GSK_PKIS: CHEK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Death-associated protein kinase 1	Inhibition	=	-2.81	%	GSK_PKIS: DAPK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase DCLK2	Inhibition	=	-0.03	%	GSK_PKIS: DCAMKL2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 2	Inhibition	=	-0.48	%	GSK_PKIS: MAPKAPK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 3	Inhibition	=	-2.07	%	GSK_PKIS: MAPKAPK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MARK1	Inhibition	=	6.09	%	GSK_PKIS: MARK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase c-TAK1	Inhibition	=	3.88	%	GSK_PKIS: MARK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP/microtubule affinity-regulating kinase 4	Inhibition	=	4.83	%	GSK_PKIS: MARK4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Maternal embryonic leucine zipper kinase	Inhibition	=	-4.7	%	GSK_PKIS: MELK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-interacting serine/threonine-protein kinase MNK1	Inhibition	=	16.5	%	GSK_PKIS: MKNK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase signal-integrating kinase 2	Inhibition	=	13.69	%	GSK_PKIS: MNK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP/microtubule affinity-regulating kinase 2	Inhibition	=	4.05	%	GSK_PKIS: PAR-1Balpha mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
PAS domain-containing serine/threonine-protein kinase	Inhibition	=	4.15	%	GSK_PKIS: PASK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Phosphorylase kinase gamma subunit 1	Inhibition	=	2.55	%	GSK_PKIS: PHKG1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Phosphorylase kinase gamma subunit 2	Inhibition	=	6.48	%	GSK_PKIS: PHKG2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM1	Inhibition	=	-0.03	%	GSK_PKIS: PIM1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM2	Inhibition	=	-3.43	%	GSK_PKIS: PIM2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PIM3	Inhibition	=	6.5	%	GSK_PKIS: PIM3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase-activated protein kinase 5	Inhibition	=	2.56	%	GSK_PKIS: PRAK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SIK1	Inhibition	=	12.03	%	GSK_PKIS: SNF1LK (SIK) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SIK2	Inhibition	=	34.08	%	GSK_PKIS: SNF1LK2 (QIK) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase TBK1	Inhibition	=	2.56	%	GSK_PKIS: TBK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Testis-specific serine/threonine-protein kinase 1	Inhibition	=	5.32	%	GSK_PKIS: TSSK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Testis-specific serine/threonine-protein kinase 2	Inhibition	=	4.98	%	GSK_PKIS: TSSK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I alpha	Inhibition	=	0.8	%	GSK_PKIS: CK1a mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I gamma 1	Inhibition	=	-4.26	%	GSK_PKIS: CK1-g1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I gamma 2	Inhibition	=	-5.36	%	GSK_PKIS: CK1-g2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Casein kinase I isoform gamma-3	Inhibition	=	-3.3	%	GSK_PKIS: CK1-g3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 1	Inhibition	=	0.55	%	GSK_PKIS: CDK1/cyclinB mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 2	Inhibition	=	8.02	%	GSK_PKIS: CDK2/cyclinA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 2	Inhibition	=	-2.32	%	GSK_PKIS: CDK2/cyclinE mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
CDK3/Cyclin E	Inhibition	=	0.9	%	GSK_PKIS: CDK3/cyclinE mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 4	Inhibition	=	-4.27	%	GSK_PKIS: CDK4/cyclinD mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 5	Inhibition	=	-0.49	%	GSK_PKIS: CDK5/p35 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Cyclin-dependent kinase 6	Inhibition	=	-8.82	%	GSK_PKIS: CDK6/cyclinD3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase CLK2	Inhibition	=	5.72	%	GSK_PKIS: CLK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase CLK3	Inhibition	=	-2.92	%	GSK_PKIS: CLK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Inhibition	=	2.17	%	GSK_PKIS: DYRK1A mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Inhibition	=	-0.65	%	GSK_PKIS: DYRK1B mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual-specificity tyrosine-phosphorylation regulated kinase 2	Inhibition	=	2.96	%	GSK_PKIS: DYRK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Glycogen synthase kinase-3 alpha	Inhibition	=	34.68	%	GSK_PKIS: GSK3A mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Glycogen synthase kinase-3 beta	Inhibition	=	32.38	%	GSK_PKIS: GSK3B mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Homeodomain-interacting protein kinase 1	Inhibition	=	-0.32	%	GSK_PKIS: HIPK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Homeodomain-interacting protein kinase 4	Inhibition	=	3.74	%	GSK_PKIS: HIPK4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
c-Jun N-terminal kinase 2	Inhibition	=	-0.57	%	GSK_PKIS: JNK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase ERK2	Inhibition	=	-0.07	%	GSK_PKIS: MAPK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase ERK1	Inhibition	=	2.27	%	GSK_PKIS: MAPK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SRPK3	Inhibition	=	0.28	%	GSK_PKIS: MSSK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 alpha	Inhibition	=	-0.98	%	GSK_PKIS: P38alpha mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 beta	Inhibition	=	0.89	%	GSK_PKIS: P38beta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 delta	Inhibition	=	-2.04	%	GSK_PKIS: P38delta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
MAP kinase p38 gamma	Inhibition	=	-1.27	%	GSK_PKIS: P38gamma mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase SRPK1	Inhibition	=	4.2	%	GSK_PKIS: SRPK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
PI3-kinase p110-alpha subunit	Inhibition	=	-3.79	%	GSK_PKIS: PI3K-alpha mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
PI3-kinase p110-delta subunit	Inhibition	=	-2.3	%	GSK_PKIS: PI3K-delta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
PI4-kinase beta subunit	Inhibition	=	-1.85	%	GSK_PKIS: PI4K-beta mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Sphingosine kinase 1	Inhibition	=	0.02	%	GSK_PKIS: SPHK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Sphingosine kinase 2	Inhibition	=	-0.25	%	GSK_PKIS: SPHK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Casein kinase II alpha	Inhibition	=	10.75	%	GSK_PKIS: CK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase alpha subunit	Inhibition	=	-1.74	%	GSK_PKIS: IKKA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase beta subunit	Inhibition	=	3.32	%	GSK_PKIS: IKKB mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase epsilon subunit	Inhibition	=	4.51	%	GSK_PKIS: IKKE mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Nek1	Inhibition	=	9.07	%	GSK_PKIS: NEK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK2	Inhibition	=	-1.3	%	GSK_PKIS: NEK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK6	Inhibition	=	2.69	%	GSK_PKIS: NEK6 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK7	Inhibition	=	-2.76	%	GSK_PKIS: NEK7 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase NEK9	Inhibition	=	5.21	%	GSK_PKIS: NEK9 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PLK1	Inhibition	=	-0.54	%	GSK_PKIS: PLK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual specificity protein kinase TTK	Inhibition	=	5.77	%	GSK_PKIS: TTK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-A	Inhibition	=	13.0	%	GSK_PKIS: Aurora-A mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-B	Inhibition	=	7.54	%	GSK_PKIS: Aurora-B mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase Aurora-C	Inhibition	=	-1.49	%	GSK_PKIS: Aurora-C mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase 10	Inhibition	=	16.32	%	GSK_PKIS: LOK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Mitogen-activated protein kinase kinase kinase kinase 2	Inhibition	=	1.25	%	GSK_PKIS: MAP4K2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Mitogen-activated protein kinase kinase kinase kinase 4	Inhibition	=	16.89	%	GSK_PKIS: MAP4K4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Dual specificity mitogen-activated protein kinase kinase 1	Inhibition	=	-0.71	%	GSK_PKIS: MEK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Misshapen-like kinase 1	Inhibition	=	16.85	%	GSK_PKIS: MINK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST1	Inhibition	=	7.14	%	GSK_PKIS: MST1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST2	Inhibition	=	7.42	%	GSK_PKIS: MST2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase MST4	Inhibition	=	-2.88	%	GSK_PKIS: MST4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 1	Inhibition	=	1.58	%	GSK_PKIS: PAK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 2	Inhibition	=	-0.99	%	GSK_PKIS: PAK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK 3	Inhibition	=	0.31	%	GSK_PKIS: PAK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK7	Inhibition	=	10.85	%	GSK_PKIS: PAK5 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase PAK6	Inhibition	=	3.44	%	GSK_PKIS: PAK6 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	80.15	%	GSK_PKIS: ABL1 (E255K mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	87.14	%	GSK_PKIS: ABL1 (H396P mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	88.06	%	GSK_PKIS: ABL1 (M351T mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	84.24	%	GSK_PKIS: ABL1 (Q252H mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	28.49	%	GSK_PKIS: ABL1 (T315I mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	85.3	%	GSK_PKIS: ABL1 (Y253F mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL	Inhibition	=	72.16	%	GSK_PKIS: ABL1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
ALK tyrosine kinase receptor	Inhibition	=	-4.64	%	GSK_PKIS: ALK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ABL2	Inhibition	=	59.45	%	GSK_PKIS: ARG mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor UFO	Inhibition	=	-2.08	%	GSK_PKIS: AXL mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BLK	Inhibition	=	15.75	%	GSK_PKIS: BLK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BMX	Inhibition	=	16.12	%	GSK_PKIS: BMX mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BRK	Inhibition	=	15.2	%	GSK_PKIS: BRK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase BTK	Inhibition	=	-2.79	%	GSK_PKIS: BTK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase CSK	Inhibition	=	7.17	%	GSK_PKIS: CSK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Discoidin domain-containing receptor 2	Inhibition	=	1.99	%	GSK_PKIS: DDR2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	8.31	%	GSK_PKIS: EGFR mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	30.83	%	GSK_PKIS: EGFR (L858R mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	10.62	%	GSK_PKIS: EGFR (L861Q mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	5.78	%	GSK_PKIS: EGFR (T790M mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Epidermal growth factor receptor erbB1	Inhibition	=	6.65	%	GSK_PKIS: EGFR (T790M-L858R mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 2	Inhibition	=	0.55	%	GSK_PKIS: EPHA2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 3	Inhibition	=	-0.79	%	GSK_PKIS: EPHA3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-A receptor 4	Inhibition	=	25.6	%	GSK_PKIS: EPHA4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 2	Inhibition	=	16.21	%	GSK_PKIS: EPHB2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 3	Inhibition	=	-4.51	%	GSK_PKIS: EPHB3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Ephrin type-B receptor 4	Inhibition	=	0.65	%	GSK_PKIS: EPHB4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Receptor protein-tyrosine kinase erbB-2	Inhibition	=	7.49	%	GSK_PKIS: ERBB2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Receptor protein-tyrosine kinase erbB-4	Inhibition	=	2.45	%	GSK_PKIS: ERBB4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FER	Inhibition	=	4.82	%	GSK_PKIS: FER mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FES	Inhibition	=	-1.27	%	GSK_PKIS: FES mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 1	Inhibition	=	-2.61	%	GSK_PKIS: FGFR1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 2	Inhibition	=	10.7	%	GSK_PKIS: FGFR2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 3	Inhibition	=	3.63	%	GSK_PKIS: FGFR3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Fibroblast growth factor receptor 4	Inhibition	=	-3.96	%	GSK_PKIS: FGFR4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FGR	Inhibition	=	18.99	%	GSK_PKIS: FGR mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 1	Inhibition	=	1.4	%	GSK_PKIS: FLT1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor FLT3	Inhibition	=	6.95	%	GSK_PKIS: FLT3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor FLT3	Inhibition	=	9.6	%	GSK_PKIS: FLT3 (D835Y mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 3	Inhibition	=	-4.88	%	GSK_PKIS: FLT4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Macrophage colony stimulating factor receptor	Inhibition	=	24.9	%	GSK_PKIS: FMS mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FYN	Inhibition	=	25.58	%	GSK_PKIS: FYN mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase HCK	Inhibition	=	16.31	%	GSK_PKIS: HCK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Insulin-like growth factor I receptor	Inhibition	=	-8.19	%	GSK_PKIS: IGF1R mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Insulin receptor	Inhibition	=	-4.12	%	GSK_PKIS: INSR mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Insulin receptor-related protein	Inhibition	=	0.57	%	GSK_PKIS: IRR mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ITK/TSK	Inhibition	=	-1.27	%	GSK_PKIS: ITK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK1	Inhibition	=	16.28	%	GSK_PKIS: JAK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK2	Inhibition	=	0.37	%	GSK_PKIS: JAK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase JAK3	Inhibition	=	-2.19	%	GSK_PKIS: JAK3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Vascular endothelial growth factor receptor 2	Inhibition	=	11.2	%	GSK_PKIS: KDR mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	83.36	%	GSK_PKIS: KIT mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	3.79	%	GSK_PKIS: KIT (D816V mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	6.36	%	GSK_PKIS: KIT (T6701 mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Stem cell growth factor receptor	Inhibition	=	18.75	%	GSK_PKIS: KIT (V560G mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase LCK	Inhibition	=	29.31	%	GSK_PKIS: LCK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Leukocyte tyrosine kinase receptor	Inhibition	=	0.9	%	GSK_PKIS: LTK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Lyn	Inhibition	=	47.25	%	GSK_PKIS: LYN A (splice variant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Lyn	Inhibition	=	41.63	%	GSK_PKIS: LYN B (splice variant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Proto-oncogene tyrosine-protein kinase MER	Inhibition	=	4.47	%	GSK_PKIS: MER mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Hepatocyte growth factor receptor	Inhibition	=	6.87	%	GSK_PKIS: MET mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Muscle, skeletal receptor tyrosine protein kinase	Inhibition	=	17.06	%	GSK_PKIS: MUSK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	53.62	%	GSK_PKIS: PDGFRA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	45.61	%	GSK_PKIS: PDGFRA (D842V mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	18.33	%	GSK_PKIS: PDGFRA (T674I mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor alpha	Inhibition	=	50.95	%	GSK_PKIS: PDGFRA (V561D mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Platelet-derived growth factor receptor beta	Inhibition	=	49.91	%	GSK_PKIS: PDGFRB mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase FRK	Inhibition	=	0.9	%	GSK_PKIS: PTK5 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Protein tyrosine kinase 2 beta	Inhibition	=	10.54	%	GSK_PKIS: PYK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	13.94	%	GSK_PKIS: RET mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	12.54	%	GSK_PKIS: RET (V804L mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor RET	Inhibition	=	32.84	%	GSK_PKIS: RET (Y791F mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Macrophage-stimulating protein receptor	Inhibition	=	0.14	%	GSK_PKIS: RON mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Proto-oncogene tyrosine-protein kinase ROS	Inhibition	=	4.38	%	GSK_PKIS: ROS mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase SRC	Inhibition	=	50.4	%	GSK_PKIS: SRC mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase Srms	Inhibition	=	6.19	%	GSK_PKIS: SRMS mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase SYK	Inhibition	=	-1.09	%	GSK_PKIS: SYK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TEC	Inhibition	=	5.03	%	GSK_PKIS: TEC mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TIE-2	Inhibition	=	9.67	%	GSK_PKIS: TIE2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Non-receptor tyrosine-protein kinase TNK1	Inhibition	=	19.33	%	GSK_PKIS: TNK1 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine kinase non-receptor protein 2	Inhibition	=	3.07	%	GSK_PKIS: TNK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Nerve growth factor receptor Trk-A	Inhibition	=	7.04	%	GSK_PKIS: TRKA mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Neurotrophic tyrosine kinase receptor type 2	Inhibition	=	6.69	%	GSK_PKIS: TRKB mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
NT-3 growth factor receptor	Inhibition	=	9.77	%	GSK_PKIS: TRKC mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TXK	Inhibition	=	4.69	%	GSK_PKIS: TXK mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase TYK2	Inhibition	=	3.46	%	GSK_PKIS: TYK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase receptor TYRO3	Inhibition	=	4.59	%	GSK_PKIS: TYRO3 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase YES	Inhibition	=	36.37	%	GSK_PKIS: YES mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Tyrosine-protein kinase ZAP-70	Inhibition	=	-3.33	%	GSK_PKIS: ZAP70 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase B-raf	Inhibition	=	-1.09	%	GSK_PKIS: BRAF mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase B-raf	Inhibition	=	-0.68	%	GSK_PKIS: BRAF (V599E mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Serine/threonine-protein kinase RAF	Inhibition	=	-4.3	%	GSK_PKIS: CRAF mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Interleukin-1 receptor-associated kinase 4	Inhibition	=	0.01	%	GSK_PKIS: IRAK4 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Leucine-rich repeat serine/threonine-protein kinase 2	Inhibition	=	7.17	%	GSK_PKIS: LRRK2 mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Leucine-rich repeat serine/threonine-protein kinase 2	Inhibition	=	18.11	%	GSK_PKIS: LRRK2 (G2019S mutant) mean inhibition at 1 uM [Nanosyn]	CHEMBL1961873
Inhibitor of nuclear factor kappa B kinase alpha subunit	Inhibition	=	2.0	%	GSK_PKIS: IKK-alpha % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Inhibitor of nuclear factor kappa B kinase alpha subunit	Inhibition	=	-3.0	%	GSK_PKIS: IKK-alpha % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Inhibitor of nuclear factor kappa B kinase beta subunit	Inhibition	=	-3.0	%	GSK_PKIS: IKK-beta % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Inhibitor of nuclear factor kappa B kinase beta subunit	Inhibition	=	4.0	%	GSK_PKIS: IKK-beta % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Inhibitor of nuclear factor kappa B kinase epsilon subunit	Inhibition	=	1.0	%	GSK_PKIS: IKK-epsilon % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Inhibitor of nuclear factor kappa B kinase epsilon subunit	Inhibition	=	0.0	%	GSK_PKIS: IKK-epsilon % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Proto-oncogene tyrosine-protein kinase MER	Inhibition	=	-4.0	%	GSK_PKIS: Mer Kinase % inhibition at 10 uM [UNC Frye lab]	CHEMBL2007661
Unchecked	Inhibition	=	10.0	%	GSK_PKIS: PIP5K1 (Caliper assay) % inhibition at 5 uM [UNC Frye lab]	CHEMBL2007661
Serine/threonine-protein kinase TBK1	Inhibition	=	4.0	%	GSK_PKIS: TBK1 % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Serine/threonine-protein kinase TBK1	Inhibition	=	-1.0	%	GSK_PKIS: TBK1 % inhibition at 1 uM [UNC Frye lab]	CHEMBL2007661
Renilla-luciferin 2-monooxygenase	AC50	=		nM	GSK_PKIS: Inhibition of Sea Pansy Luciferase (Data from PubChem: AID 652015) [NIH NCATS]	CHEMBL2303647
Luciferin 4-monooxygenase	AC50	=	16343.2	nM	GSK_PKIS: Inhibition of Firefly Luciferase (Data from PubChem: AID 652016) [NIH NCATS]	CHEMBL2303647