NA-DB

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	Compound ID	Cluster 2	Compound Type ALL-match Base-match Ribose-match	Target/Cell	Structure	Activity				Assay Description	Source
	Compound ID	Cluster 2	Compound Type ALL-match Base-match Ribose-match	Target/Cell	Structure	Type Ki Other	Relation =	Value	Unit nM None	Assay Description	Source
	NAs.000015	2	all-match	Adenosine A1 receptor		Ki	=	95.0	nM	Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells	CHEMBL1142938
	NAs.000015	2	all-match	Adenosine A2a receptor		Ki	=	758.0	nM	Displacement of [3H]NECA from human recombinant adenosine A2A receptor expressed in CHO cells	CHEMBL1142938
	NAs.000015	2	all-match	Adenosine A3 receptor		Ki	=	5.4	nM	Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cells	CHEMBL1142938
	NAs.000015	2	all-match	Adenosine receptors; A1 & A3		Other	=	18.0	None	Selectivity for human adenosine A3 receptor over human adenosine A1 receptor	CHEMBL1142938
	NAs.000015	2	all-match	Adenosine receptors; A2a & A3		Other	=	140.0	None	Selectivity for human adenosine A3 receptor over human adenosine A2A receptor	CHEMBL1142938