Showing 1 to 7 of 7 entries Per page:
Compound ID
Cluster
Compound Type
Target/Cell Structure Activity Assay Description Source
Type
Relation
Value
Unit
NAs.000026 2 ribose-match Adenosine A3 receptor NAs.000026 Ki = 41.0 nM Displacement of [125I]-AB MECA from recombinant human adenosine A3 receptor expressed in HEK cells CHEMBL1138752
NAs.000026 2 ribose-match Adenosine A1 receptor NAs.000026 Ki = 3700.0 nM Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cells CHEMBL1138752
NAs.000026 2 ribose-match Adenosine A2a receptor NAs.000026 Ki = 4000.0 nM Displacement of [3H]CGS-21680 from recombinant human adenosine A2a receptor expressed in HEK cells CHEMBL1138752
NAs.000026 2 ribose-match Adenosine receptors; A1 & A3 NAs.000026 Other = 90.0 None Ratio of binding to adenosine A1 and adenosine A3 receptor CHEMBL1138752
NAs.000026 2 ribose-match Adenosine receptors; A2a & A3 NAs.000026 Other = 100.0 None Ratio of binding to adenosine A2a and adenosine A3 receptor CHEMBL1138752
NAs.000026 2 ribose-match Adenosine A1 receptor NAs.000026 Ki = 3700.0 nM Displacement of [3H]CPX from adenosine A1 receptor in DDT membranes CHEMBL1146258
NAs.000026 2 ribose-match Adenosine A3 receptor NAs.000026 Ki = 41.0 nM Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cells CHEMBL1146258