NA-DB

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	Compound ID	Cluster 2	Compound Type ALL-match Base-match Ribose-match	Target/Cell	Structure	Activity				Assay Description	Source
	Compound ID	Cluster 2	Compound Type ALL-match Base-match Ribose-match	Target/Cell	Structure	Type Ki EC50 Other	Relation = >	Value	Unit nM % None	Assay Description	Source
	NAs.000027	2	ribose-match	Adenosine A1 receptor		Ki	=	8.5	nM	Displacement of [3H]CHA from human adenosine A1 receptor expressed in CHO cells	CHEMBL1142924
	NAs.000027	2	ribose-match	Adenosine A2b receptor		EC50	=	7.3	nM	Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP production	CHEMBL1142924
	NAs.000027	2	ribose-match	Adenosine A3 receptor		Ki	=	38.4	nM	Displacement of [3H]ABMECA from human adenosine A3 receptor expressed in CHO cells	CHEMBL1142924
	NAs.000027	2	ribose-match	Adenosine A2a receptor		Ki	>	1000.0	nM	Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells	CHEMBL1142924
	NAs.000027	2	ribose-match	Adenosine A2a receptor		Other	=	45.0	%	Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells	CHEMBL1142924
	NAs.000027	2	ribose-match	Adenosine A2b receptor		Other	=	-0.863	None	Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of adenylate cyclase	CHEMBL1145544
	NAs.000027	2	ribose-match	Adenosine A2b receptor		Other	=	1.327	None	Agonist activity human adenosine A2B receptor expressed in CHO cells assessed as stimulation of adenylate cyclase relative to NECA	CHEMBL1145544