| Compound ID |
Cluster
|
Compound Type
|
Target/Cell | Structure | Activity | Assay Description | Source | ||||
|---|---|---|---|---|---|---|---|---|---|---|---|
|
Type
|
Relation
|
Value
|
Unit
|
||||||||
| NAs.000054 | 7 | all-match | Adenosine A1 receptor |  |
Ki | = | 20000.0 | nM | Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells | CHEMBL1153377 | |
| NAs.000054 | 7 | all-match | Adenosine A2a receptor | |
Ki | = | 12000.0 | nM | Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cells | CHEMBL1153377 | |
| NAs.000054 | 7 | all-match | Adenosine A2b receptor | |
Ki | > | 30000.0 | nM | Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activity | CHEMBL1153377 | |
| NAs.000054 | 7 | all-match | Adenosine A3 receptor | |
Ki | > | 100000.0 | nM | Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cells | CHEMBL1153377 | |