显示 1 到 50 条，共 159 条数据 每页数据量:
Compound ID
Cluster
Compound Type
Target Name Img Activity Assay Description Source
Type
Relation
Value
Unit
NAs.000040 7 ribose-match Adenosine receptor A2a and A3 NAs.000040 Ratio = 0.07 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000044 2 ribose-match Adenosine receptor A2a and A3 NAs.000044 Ratio = 27.0 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000059 7 all-match Adenosine receptor A2a and A3 NAs.000059 Ratio = 0.66 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000117 8 ribose-match Adenosine receptor A2a and A3 NAs.000117 Ratio = 4.7 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000192 2 ribose-match Adenosine receptor A2a and A3 NAs.000192 Selectivity = 140.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000304 2 ribose-match Adenosine receptor A2a and A3 NAs.000304 Ratio = 1.5 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000305 2 ribose-match Adenosine receptor A2a and A3 NAs.000305 Ratio = 34.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000306 2 ribose-match Adenosine receptor A2a and A3 NAs.000306 Ratio > 140.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000309 8 ribose-match Adenosine receptor A2a and A3 NAs.000309 Ratio > 50.0 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000336 7 all-match Adenosine receptor A2a and A3 NAs.000336 Ratio = 5.5 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000359 2 ribose-match Adenosine receptor A2a and A3 NAs.000359 Ratio = 0.046 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000403 2 all-match Adenosine receptor A2a and A3 NAs.000403 Ratio = 0.033 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000448 2 ribose-match Adenosine receptor A2a and A3 NAs.000448 Selectivity = 58.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000494 2 ribose-match Adenosine receptor A2a and A3 NAs.000494 Ratio = 18.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000517 7 all-match Adenosine receptor A2a and A3 NAs.000517 Ratio = 0.046 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000521 7 all-match Adenosine receptor A2a and A3 NAs.000521 Ratio = 0.068 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000598 2 ribose-match Adenosine receptor A2a and A3 NAs.000598 Ratio = 2.6 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000617 2 all-match Adenosine receptor A2a and A3 NAs.000617 Selectivity = 0.07 None Selectivity towards Adenosine A3 receptor to Adenosine A2A receptor CHEMBL1135881
NAs.000617 2 all-match Adenosine receptor A2a and A3 NAs.000617 Ratio = 1.9 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000627 2 all-match Adenosine receptor A2a and A3 NAs.000627 Selectivity > 2.9 None Selectivity towards Adenosine A3 receptor to Adenosine A2A receptor CHEMBL1135881
NAs.000628 2 ribose-match Adenosine receptor A2a and A3 NAs.000628 Ratio = 1400.0 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000659 2 ribose-match Adenosine receptor A2a and A3 NAs.000659 Ratio = 19.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000688 2 ribose-match Adenosine receptor A2a and A3 NAs.000688 Selectivity = 0.13 None Selectivity towards Adenosine A3 receptor to Adenosine A2A receptor CHEMBL1135881
NAs.000701 7 all-match Adenosine receptor A2a and A3 NAs.000701 Ratio = 0.08 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000734 2 ribose-match Adenosine receptor A2a and A3 NAs.000734 Ratio = 1.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000749 2 ribose-match Adenosine receptor A2a and A3 NAs.000749 Ratio = 11.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000808 2 ribose-match Adenosine receptor A2a and A3 NAs.000808 Selectivity = 510.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000832 2 ribose-match Adenosine receptor A2a and A3 NAs.000832 Ratio > 300.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000862 2 ribose-match Adenosine receptor A2a and A3 NAs.000862 Selectivity = 11.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000868 2 ribose-match Adenosine receptor A2a and A3 NAs.000868 Selectivity = 190.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000879 2 all-match Adenosine receptor A2a and A3 NAs.000879 Ratio = 4.0 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000900 2 ribose-match Adenosine receptor A2a and A3 NAs.000900 Selectivity = 96.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000906 2 ribose-match Adenosine receptor A2a and A3 NAs.000906 Ratio = 1400.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000915 2 ribose-match Adenosine receptor A2a and A3 NAs.000915 Ratio = 3.8 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000938 2 ribose-match Adenosine receptor A2a and A3 NAs.000938 Ratio = 0.026 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000952 2 all-match Adenosine receptor A2a and A3 NAs.000952 Ratio = 0.0091 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000954 2 ribose-match Adenosine receptor A2a and A3 NAs.000954 Ratio Ki = 51.0 None Selectivity ratio of Ki for rat adenosine A2A receptor to Ki for rat adenosine A3 receptor expressed in CHO cells CHEMBL2177029
NAs.000954 2 ribose-match Adenosine receptor A2a and A3 NAs.000954 Ratio = 51.0 None Ratio of Ki for A2a and A3 receptors CHEMBL1127377
NAs.000954 2 ribose-match Adenosine receptor A2a and A3 NAs.000954 Ratio = 51.0 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.000954 2 ribose-match Adenosine receptor A2a and A3 NAs.000954 Selectivity = 51.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000954 2 ribose-match Adenosine receptor A2a and A3 NAs.000954 Ratio = 51.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000959 2 ribose-match Adenosine receptor A2a and A3 NAs.000959 Ratio > 4000.0 None Selectivity for binding affinity towards A2A adenosine receptor in rat striatal membrane and rat A3 receptor expressed in CHO cells. CHEMBL1131059
NAs.000967 2 all-match Adenosine receptor A2a and A3 NAs.000967 Selectivity = 1.9 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.000970 2 ribose-match Adenosine receptor A2a and A3 NAs.000970 Selectivity = 0.07 None Selectivity towards Adenosine A3 receptor to Adenosine A2A receptor CHEMBL1135881
NAs.000993 2 ribose-match Adenosine receptor A2a and A3 NAs.000993 Selectivity < 1.0 None Selectivity towards Adenosine A3 receptor to Adenosine A2A receptor CHEMBL1135881
NAs.001001 8 ribose-match Adenosine receptor A2a and A3 NAs.001001 Ratio = 5.5 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.001002 2 ribose-match Adenosine receptor A2a and A3 NAs.001002 Selectivity = 13.0 None Selectivity, ratio between A2A receptor binding affinity / A3 receptor binding affinity CHEMBL1129034
NAs.001006 7 all-match Adenosine receptor A2a and A3 NAs.001006 Ratio = 0.18 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362
NAs.001014 2 ribose-match Adenosine receptor A2a and A3 NAs.001014 Ratio Ki = 7.2 None Selectivity ratio of Ki for rat adenosine A2A receptor to Ki for rat adenosine A3 receptor expressed in CHO cells CHEMBL2177029
NAs.001016 8 ribose-match Adenosine receptor A2a and A3 NAs.001016 Ratio > 7.0 None Ratio of the binding affinities against rat brain A2a and A3 receptors, KiA2a/KiA3. CHEMBL1128362